Discovery of the Potent, Selective, Orally Available CXCR7 Antagonist ACT- 1004-1239 | Journal of Medicinal Chemistry
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ACT‐1004‐1239, a first‐in‐class CXCR7 antagonist with both immunomodulatory and promyelinating effects for the treatment of inflammatory demyelinating diseases - Pouzol - 2021 - The FASEB Journal - Wiley Online Library
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Frontiers | Absorption, Metabolism, and Excretion of ACT-1004-1239, a First-In-Class CXCR7 Antagonist: In Vitro, Preclinical, and Clinical Data
![Treatment with ACT-1004-1239 dose-dependently increases plasma CXCL11... | Download Scientific Diagram Treatment with ACT-1004-1239 dose-dependently increases plasma CXCL11... | Download Scientific Diagram](https://www.researchgate.net/publication/362353923/figure/fig17/AS:1183535062880320@1659188156350/Treatment-with-ACT-1004-1239-dose-dependently-increases-plasma-CXCL11-and-CXCL12-levels.png)
Treatment with ACT-1004-1239 dose-dependently increases plasma CXCL11... | Download Scientific Diagram
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Preclinical development of ACT-1004-1239, a potent and selective CXCR7/ACKR3 antagonist in multiple sclerosis treatment
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Discovery of the Potent, Selective, Orally Available CXCR7 Antagonist ACT- 1004-1239 | Journal of Medicinal Chemistry
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Target engagement of the first-in-class CXCR7 antagonist ACT-1004-1239 following multiple-dose administration in mice and humans - ScienceDirect
Preclinical development of ACT-1004-1239, a potent and selective CXCR7/ACKR3 antagonist in multiple sclerosis treatment
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